Antimalarial Activity of C-10 Substituted Triazolyl Artemisinin

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참고문헌 (27)

1. Klayman DL, "Qinghaosu(artemisinin) : an antimalarial drug from China", Science, 228, pp.1049~1055 (1985)
2. Lee S, "Artemisinin, promising lead natural product for various drug developments", Mini Rev Med Chem, 7, pp.411~422 (2007)
3. Luo XD, "The chemistry, pharmacology, and clinical applications of qinghaosu (artemisinin) and its derivatives", Med Res Rev, 7, pp.29~52 (1987)
4. Jung M, "Current developments in the chemistry of artemisinin and related compounds", Curr Med Chem, 1, pp.35~49 (1994)
5. Haynes RK, "From Qinghao, marvelous herb of antiquity, to the antimalarial trioxane qinghaosu-and some remarkable new chemistry", Acc Chem Res, 30, pp.73~79 (1997)
6. Vroman JA, "Current progress in the chemistry, medicinal chemistry and drug design of artemisinin based antimalarials", Curr Pharm Design, 5, pp.101~138 (1999)
7. Beekman AC, "Stereochemistry-dependent cytotoxicity of some artemisinin derivatives", J Nat Prod, 60, pp.325~330 (1997)
8. Jung M, "Antitumor activity of novel deoxoartemisinin monomers, dimers, and trimer", J Med Chem, 46, pp.987~994 (2003)
9. Posner GH, "Orally active, antimalarial, anticancer, artemisinin-derived trioxane dimers with high stability and efficacy", J Med Chem, 46, pp.1060~1065 (2003)
10. Brewer TG, "Neurotoxicity in animals due to arteether and artemether", Trans R Soc Trop Med Hyg, 88, pp.33~36 (1994)
11. Lin AJ, "Antimalarial activity of new watersoluble dihydroartemisinin derivatives. 2. Stereospecificity of the ether side chain", J Med Chem, 32, pp.1249~1252 (1989)
12. Lin AJ, "Antimalarial activity of new water-soluble dihydroartemisinin derivatives", J Med Chem, 30, pp.2147~2150 (1987)
13. Lin AJ, "Antimalarial activity of new dihydroartemisinin derivatives. 6. alpha-Alkylbenzylic ethers", J Med Chem, 38, pp.764~770 (1995)
14. Jung M, "A short and stereospecific synthesis of (+)-deoxoartemisinin and (-)-deoxodesoxyartemisinin", Tetrahedron Lett, 44, pp.5973~5976 (1989)
15. Jung M, "Synthesis and antimalarial activity of (+)-deoxoartemisinin", J Med Chem, 33, pp.1516~1518 (1990)
16. 이석준, "Antimalarial activity of thiophenyl- and benzenesulfonyl-dihydroartemisinin", The Korean Journal of Parasitology, 43(3), pp.123~126 (2005), 대한기생충학ㆍ열대의학회
17. Jung M, "Stability of acetal and non acetal-type analogs of artemisinin in simulated stomach acid", Bioorg Med Chem Lett, 8, pp.1003~1006 (1998)
18. Gordi T, "Artemisinin derivatives: toxic for laboratory animals, safe for humans?", Toxicol Lett, 147, pp.99~107 (2004)
19. Haynes RK, "Preparation of N-sulfonyl- and N-carbonyl-11-azaartemisinins with greatly enhanced thermal stabilities: in vitro antimalarial activities", Chem Med Chem, 2, pp.1464~1479 (2007)
20. Haynes RK, "Artemisone--a highly active antimalarial drug of the artemisinin class", Angew Chem Int Ed Engl, 45, pp.2082~2088 (2006)
21. Cho S, "Synthesis of 10-substituted triazolyl artemisinins possessing anticancer activity via Huisgen 1,3-dipolar cycloaddition", Bioorg Med Chem Lett, 19, pp.382~385 (2009)
22. Oh S, "Acid-catalyzed synthesis of 10-substituted triazolyl artemisinins and their growth inhibitory activity against various cancer cells", Bioorg Med Chem Lett, 20, pp.4112~4115 (2010)
23. 이석준, "Synthesis of 10β-Substituted Triazolyl Artemisinins and Their Growth Inhibitory Activity against Various Cancer Cells", Bulletin of the Korean Chemical Society, 32(2), pp.737~740 (2011), 대한화학회
24. Nguyen-Dinh P, "Plasmodium falciparum in vitro : determination of chloroquine sensitivity of three new strains by a modified 48-hour test", Am J Trop Med Hyg, 29, pp.339~342 (1980)
25. Jensen JB, "Plasmodium falciparum in culture : establishment of additional strains", Am J Trop Med Hyg, 27, pp.743~746 (1978)
26. Desjardins RE, "Quantitative assessment of antimalarial activity in vitro by a semiautomated microdilution technique", Antimicrob Agents Chemother, 16, pp.710~718 (1979)
27. Delhaes L, "Synthesis of ferroquine enantiomers: first investigation of effects of metallocenic chirality upon antimalarial activity and cytotoxicity", Chembiochem, 3, pp.418~423 (2002)

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