본문 바로가기
KERD
논문KCI 등재

An Improved Procedure for the Synthesis of 1,5-Benzothiazepines Using Ceric Ammonium Nitrate (CAN)

Asha V. Chate|Ratnadeep S. Joshi|Priyanka G. Mandhane|Charansingh H. Gill
대한화학회|2011.10|대한화학회지 (Journal of the Korean Chemical Society)|제55권 제5호|pp. 776-780

2

조회

0

다운로드

2

인용

0

참고문헌

키워드

1CatalysisCAN5-BenzothiazepineChalconeUltrasound irradiation
주제분류화학

초록

A mild and efficient procedure for the synthesis of various 1,5-benzothiazepines were developed. This method provides an easy access for preparation of 1,5-benzothiazepine derivatives in the presence of 10 mol% catalyst of CAN under ultrasonic irradiation. This method provided clean conversion, mild reaction condition, no use of toxic solvent and shorter reaction time compared to other reported method.

Abstract

A mild and efficient procedure for the synthesis of various 1,5-benzothiazepines were developed. This method provides an easy access for preparation of 1,5-benzothiazepine derivatives in the presence of 10 mol% catalyst of CAN under ultrasonic irradiation. This method provided clean conversion, mild reaction condition, no use of toxic solvent and shorter reaction time compared to other reported method.

참고문헌 (40)

  1. Sarro, G. D., , Eur. J. Med. Chem, 30, pp.925~ (1995)
  2. Shinichi, Y., , J. Org. Chem, 61, pp.8586~ (1996)
  3. Kurokawa, J., , Eur. J. Pharmacol, 325, pp.229~ (1997)
  4. Miyata, O., , Tetrahedron, 53, pp.2421~ (1997)
  5. Grandolini, G., , Eur. J. Med. Chem, 34, pp.701~ (1999)
  6. Yang, X., , Tetrahedron: Asymmetry, 11, pp.4447~ (2000)
  7. Urbanski, M. J., , Bioorg. Med. Chem. Lett, 13, pp.4031~ (2003)
  8. Di Santo, R., , Farmaco, 60, pp.385~ (2005)
  9. Lévai, A., , J. Heterocycl. Chem, 37, pp.199~ (2000)
  10. Kodomari, M., , Synth. Commun, 34, pp.1783~ (2004)
  11. Patel, V. M., , Indian J. Chem. Sect. B: Org. Chem. Incl. Med. Chem, 43, pp.199~ (2004)
  12. Katritzky, A. R., , J. Heterocycl. Chem, 37, pp.1655~ (2000)
  13. Dandia, A., , Green Chem, 4, pp.599~ (2002)
  14. Lévai, A., , J. Heterocycl. Chem, 41, pp.399~ (2004)
  15. Levai, A., , J. Heterocycl. Commun, 8, pp.227~ (2002)
  16. Lévai, A., , J. Heterocycl. Commun, 8, pp.375~ (2002)
  17. Micheli, F., , J. Comb. Chem, 3, pp.224~ (2001)
  18. Pant, S., , Molecules, 3, pp.159~ (1998)
  19. Upreti, M., , Indian J. Chem, 36, pp.1181~ (1997)
  20. Pant, S., , Sect. B: Indian J. Chem, 35, pp.794~ (1996)
  21. Gaplovsky, A., , J. Org. Chem, 65, pp.8444~ (2000)
  22. Suslick, K. S., "In ultrasound, it’s Chemical, physical and biological effects" (1988), VCH
  23. Rajagopal, R., , Chem. Commun, pp.616~ (2002)
  24. Deshmukh, R. R., , Chem. Commun, pp.1544~ (2001)
  25. Hwu, J. R., , Curr. Sci, 81, pp.1043~ (2001)
  26. Nair, V., , Synlett, pp.156~ (2003)
  27. Dhakshinmoorty, A., , Synlett, pp.3014~
  28. Varala, R., , Synlett, pp.1009~ (2006)
  29. Varala, R., , Synlett, pp.1549~ (2006)
  30. Nair, V., , Chem. Soc. Rev, pp.127~ (1997)
  31. Nair, V., , Acc. Chem. Res, pp.21~ (2004)
  32. Nair, V., , Chem. Rev, pp.1862~ (2007)
  33. Joshi, R. S., , Bioorg. Med. Chem. Lett, 20, pp.3721~ (2010)
  34. Jadhav, G. R., , J. Het. Chem, 45, pp.1287~ (2008)
  35. Jadhav, G. R., , Bioorg. & Med. Chem. Lett, 16, pp.6244~ (2008)
  36. Joshi, R. S., , Ultrason. Sonochem, 17, pp.298~ (2010)
  37. Mandhane, P. G., , Tett. Letts, 51, pp.1490~ (2010)
  38. Mandhane, P. G., , Tett. Lett, 51, pp.3138~ (2010)
  39. Wattanasin, S., , Synthesis, 8, pp.647~ (1980)
  40. Sharma, G., , Tetrahedron Lett, 49, pp.4269~ (2008)

관련 논문AI추천

An Improved Protocol on the Synthesis of Thiazolo[3,2-a]pyrimidine Using Ultrasonic Probe IrradiationPoh Wai Chia, Sian Hui Tan, Tse Seng Chuah대한화학회 · 대한화학회지2016 · 제60권 제4호Silica Sulfuric Acid as a Mild and Efficient Reagent for the Synthesis of 1,4-Diazepine and 1,5-Benzodiazepine DerivativesKavita, P. Joshi, Rajesh Kumar, Shalini Saingar, Y. C. Joshi대한화학회 · 대한화학회지2011 · 제55권 제4호Tetra Butyl Ammonium Chloride Catalyzed Synthesis of Substituted Benzimidazoles under Microwave ConditionsKarickal. R. Haridas, Ranjith. P. Karuvalam, Siji. M대한화학회 · 대한화학회지2010 · 제54권 제5호Ultrasound Mediated, Sodium Bisulfite Catalyzed, Solvent Free Synthesis of 6-Amino-3-methyl-4-substitued-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileDevanand B. Shinde, Jaiprakash N. Sangshetti, Sunil N. Darandale대한화학회 · 대한화학회지2012 · 제56권 제3호Microwave-Assisted and Conventional Synthesis of Benzothieno [3,2-e] [1,3,4] triazolo[4,3-c]pyrimidines: A Comparative Study안철진, Nitinkumar S. Shetty, Princia, Santhosh L. Gaonkar대한화학회 · 대한화학회지2014 · 제58권 제4호Synthesis and Characterization of 1-Benzofuran-2-yl thiadiazoles, Triazoles and Oxadiazoles by Conventional and Non-conventional MethodsAnanta D. Shinde, Bapurao B. Shingate, Bhima Y. Kale, Murlidhar S. Shingare대한화학회 · 대한화학회지2010 · 제54권 제5호

이 간행물의 다른 논문 (25건)

Statistical Study For The prediction of pKa Values of Substituted Benzaldoxime Based on Quantum Chemicals MethodsEmad A.S. Al-Hyali, Nezar A. Al-Azzawi, Faiz M.H. Al-Abadypp. 733-740Alkyl Group Dissociation During Corona Excitation of AlkylbenzenesYoung Wook Yoon, 이상국pp. 741-745Specific Binding of Nile Red to ApomyoglobinSalina A. Chowdhury, 임만호pp. 746-750Resolution of Aryl α-Aminoalkyl Ketones on a Doubly Tethered Liquid Chromatographic Chiral Stationary Phase Based on (+)-(18-Crown-6)-2,3,11,12-tetracarboxylic AcidHee Jin Kim, Kab Bong Jin, 현명호pp. 751-755Synthesis of (2-pyridyl)-Acetyl Chitosan and Its Antioxidant ActivityRong-chun Lipp. 756-759
원문 보기